Peptide APIs
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MOTS-C
MOTS-C API waxaa lagu soo saaraa xaalado adag oo GMP u eg iyadoo la adeegsanayo tignoolajiyada adag ee wejiga peptide synthesis (SPPS) si loo hubiyo tayada sare, nadiifnimada sare iyo xasilloonida sare ee cilmi baarista iyo isticmaalka daweynta.
Astaamaha Alaabta:Daahirnimada ≥ 99% (waxaa xaqiijiyay HPLC iyo LC-MS),
endotoxin hooseeya iyo ka kooban dareeraha haraaga ah,
Lagu soo saaray si waafaqsan ICH Q7 iyo borotokool la mid ah GMP,
Wuxuu gaari karaa wax soo saar ballaaran, laga bilaabo heerka milligaraam ee R&D dufcadaha ilaa heerka garaam iyo kiilooga ganacsiga sahayda. -
Ipamorelin
Ipamorelin API waxaa diyaariya heerka sare ** nidaamka isku dhafka peptide wejiga adag (SPPS)** waxaana lagu sameeyaa nadiifin adag iyo tijaabin tayo leh, oo ku habboon isticmaalka dhuumaha hore ee cilmi-baarista sayniska iyo horumarinta iyo shirkadaha dawooyinka.
Tilmaamaha alaabta waxaa ka mid ah:
Daahirnimada ≥99% (tijaabada HPLC)
Ma jiro endotoxin, dareere hadhaa ah oo hooseeya, faddarayn bir ah oo hooseeya
Bixi dukumentiyo tayo leh oo buuxa: COA, warbixinta daraasadda xasilloonida, falanqaynta spectrum nijaasta, iwm.
Heerarka garaam ~ kiiloogaraam la beddeli karo -
Pulegone
Pulegone waa ketone monoterpene si dabiici ah u dhacda oo laga helo saliidaha lagama maarmaanka ah ee noocyada reexaanta sida pennyroyal, spearmint, iyo basbaaska. Waxa loo istcimaalaa sida walax dhadhan, qayb udgoon, iyo dhex dhexaad u ah isku dhafka dawada iyo kiimikada. Our Pulegone API waxaa lagu soo saaray soo saarid la safeeyey iyo hababka sifaynta si loo hubiyo nadiifnimada sare, joogtaynta, iyo u hoggaansanaanta heerarka badbaadada iyo tayada habboon.
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Etelcalcetide
Etelcalcetide waa calcimimetic peptide synthetic ah oo loo isticmaalo daaweynta hyperparathyroidism secondary (SHPT) ee bukaanada qaba cudurka kelyaha ee raaga (CKD) ee hemodialysis. Waxay ka shaqeysaa iyada oo kicinaysa soo-dhoweynta kalsiyum-dareenka (CaSR) ee unugyada parathyroid, taas oo hoos u dhigta heerarka hoormoonka parathyroid (PTH) iyo hagaajinta dheef-shiid kiimikaadka macdanta. Etelcalcetide API ee nadiifka ah ee nadiifka ah waxaa lagu soo saaray isku-dhafka peptide-waji adag (SPPS) iyadoo la raacayo shuruudaha GMP, oo ku habboon qaababka la isku duro.
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Bremelanotide
Bremelanotide waa peptide synthetic iyo melanocortin receptor agonist loo sameeyay daawaynta rabitaanka galmada hypoactive (HSDD) ee haweenka ka horreeya menopause. Waxay u shaqeysaa iyada oo kicinaysa MC4R ee habka dhexe ee neerfayaasha si kor loogu qaado rabitaanka galmada iyo kacsiga. Bremelanotide API ee nadiifsanaanta sare leh waxaa lagu soo saaray isku-darka peptide-ka ee wejiga adag (SPPS) iyadoo la raacayo heerar tayo adag, oo ku habboon qaababka la isku duro.
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Etelcalcetide Hydrochloride
Etelcalcetide Hydrochloride waa calcimimetic-ku-saleysan peptide-ku-saleysan oo loo isticmaalo daaweynta hyperparathyroidism-ka sare (SHPT) ee bukaannada qaba cudurrada kelyaha ee daba-dheeraada (CKD) ee hemodialysis. Waxay u shaqeysaa iyada oo kicinaysa soo-dhoweynta kalsiyum-dareenka (CaSR) ee qanjidhada parathyroid, taas oo hoos u dhigta heerarka hoormoonka parathyroid (PTH) iyo hagaajinta dheelitirka calcium-phosphate. Etelcalcetide API-gayada waxa lagu soo saaray isku-darka peptide-ka saafiga ah oo sarreeya oo u hoggaansama heerarka tayada caalamiga ah ee alaabta la isku duro ee heerka-dawada.
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Desmopressin Acetate si loo daaweeyo Insipidus-ka-macaanka dhexe
Magaca: Desmopressin
Lambarka CAS: 16679-58-6
Qaaciddada molecular: C46H64N14O12S2
Miisaanka unugyada: 1069.22
Lambarka EINECS: 240-726-7
Wareeg gaar ah: D25 +85.5 ± 2° (waxaa lagu xisaabiyay peptide-ka bilaashka ah)
Cufnaanta: 1.56± 0.1 g/cm3 (La saadaaliyay)
RTECS No.: YW9000000
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Eptifibatide loogu talagalay daawaynta xanuunka wadnaha ee ba'an 188627-80-7
Magaca: Eptifibatide
Lambarka CAS: 188627-80-7
Qaaciddada molecular: C35H49N11O9S2
Miisaanka molecular: 831.96
Lambarka EINECS: 641-366-7
Cufnaanta: 1.60± 0.1 g/cm3 (La saadaaliyay)
Xaaladaha kaydinta: Waxaa lagu xidhay qalalan, ku kaydi qaboojiyaha, ka hooseeya -15°C
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Terlipressin Acetate oo loogu talagalay Dhiigbaxa Variceal Esophageal
Magaca: N-(N- (N-Glycylglycyl) glycyl) -8-L-lysinevasopressin
Lambarka CAS: 14636-12-5
Qaaciddada molecular: C52H74N16O15S2
Miisaanka unugyada: 1227.37
Lambarka EINECS: 238-680-8
Barta karkarinta: 1824.0± 65.0 °C (La saadaaliyay)
Cufnaanta: 1.46± 0.1 g/cm3 (La saadaaliyay)
Xaaladaha kaydinta: Ku hay meel mugdi ah, jawi aan fiicneyn, ku kaydi qaboojiyaha, ka hooseeya -15°C.
Isku-dhafka aysiidhka: (pKa) 9.90±0.15 (La saadaaliyay)
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Teriparatide Acetate API ee Lafo-jileeca CAS NO.52232-67-4
Teriparatide waa 34-peptide synthetic, oo ah 1-34 amino acid qayb ka mid ah hormoonka parathyroid ee bini'aadamka ee PTH, kaas oo ah bayooloji firfircoon N-terminal gobolka 84 amino acids endogenous parathyroid hormone PTH. Astaamaha difaaca jirka iyo bayooloji ee alaabtani waxay la mid yihiin kuwa hoormoonka parathyroid ee PTH iyo bovine parathyroid hormone PTH (bPTH).
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Atosiban Acetate Loo Isticmaalay Dhalashada Ka Hortagga Ah
Magaca: Atosiban
Lambarka CAS: 90779-69-4
Qaaciddada molecular: C43H67N11O12S2
Miisaanka molecular: 994.19
Lambarka EINECS: 806-815-5
Barta karkarinta: 1469.0± 65.0 °C (La saadaaliyay)
Cufnaanta: 1.254±0.06 g/cm3(La saadaaliyay)
Xaaladaha kaydinta: -20°C
Solubility: H2O: ≤100 mg/ml
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Carbetocin si ay uga hortagto foosha Uterine-ka iyo Dhiig-baxa dhalmada ka dib
Magaca: CARBETOCIN
Lambarka CAS: 37025-55-1
Qaaciddada molecular: C45H69N11O12S
Miisaanka molecular: 988.17
Lambarka EINECS: 253-312-6
Wareeg gaar ah: D -69.0° (c = 0.25 gudaha 1M acetic acid)
Barta karkarinta: 1477.9 ± 65.0 °C (La saadaaliyay)
Cufnaanta: 1.218± 0.06 g/cm3 (La saadaaliyay)
Xaaladaha kaydinta: -15°C
Foomka: budada
