oo China Paclitaxel 33069-62-4 Daawooyinka Botanical Anti-tumor ee Kansarka Ovarian-ka, Warshada Kansarka Naasaha iyo soo saarayaasha |Gentolex
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Paclitaxel 33069-62-4 Daawada Botanical-ka-Bada-hortagga ee Kansarka Ovarian-ka, Kansarka Naaska

Sharaxaad Gaaban:

Meesha dhalaalka: 213 °C

Barta karkarinta: 774.66°C (qiyaasta qallafsan)

Wareeg gaar ah: D20 -49°(methanol)

Cufnaanta: 1.0352 (qiyaas adag)

Barta iftiimaya: 9°C

Xaaladaha kaydinta: 2-8°C

Foomka: budada

Isku-dhafka aysiidhka: 11.90±0.20 (La saadaaliyay)

Midabka: Caddaan


Faahfaahinta Alaabta

Tags Product

Faahfaahinta Alaabta

Magaca Paclitaxel
Lambarka CAS 33069-62-4
qaacidada molecular C47H51NO14
Miisaanka molecular 853.92
Lambarka EINECS 608-826-9
Barta Karsan 774.66°C (La saadaaliyay)
Cufnaanta 0.200
Xaaladda kaydinta Ku dabool qallalan, ku kaydi qaboojiyaha, 2-8 ° C
Foomka Budada
Midabka Caddaan
Baakad Bac PE+Bacda aluminium

La mid ah

Paclitaxel HCL; Paclitaxel ( cayriin dabiiciga ah); Paclitaxelx; N-BENZYL-BETA-PHENYLISOSERINE ESTER;PACLITAXEL, TAXUS BREVIFOLIA;PACLITAXEL, TAXUSSPECIES;PACLITAXOL;PACLITAXEL

Saamaynta Dawaynta

Sharaxaada

Paclitaxel waa diterpenoid monomeric ah oo laga soo saaro jilif dhirta dabiiciga ah ee daawada Taxus.Baafinta Isotope waxay muujisay in paclitaxel kaliya ay ku xidhan tahay microtubules-ka polymerized oo aanu ka falcelinayn dimers tubulin-ka aan polymerized.Ka dib markii unugyadu ay soo gaadhaan paclitaxel, tiro badan oo microtubules ah ayaa ku urursan doona unugyada.Isku-ururinta microtubules-kan waxay faragelisaa shaqooyinka kala duwan ee unugyada, gaar ahaan qaybta unuggu waxay istaagtaa marxaladda mitirka waxayna xannibaysaa qaybta caadiga ah ee unugyada.Iyadoo loo marayo Ⅱ-Ⅲ cilmi-baaris caafimaad, paclitaxel waxay inta badan ku habboon tahay kansarka ugxan-sidaha iyo kansarka naasaha, sidoo kale waxay leedahay saameyn daweyn ah oo ku saabsan kansarka sambabada, kansarka mindhicirka, melanoma, kansarka madaxa iyo qoorta, lymphoma iyo burada maskaxda.

 

Tilmaamaha

Waxay saameyn wanaagsan ku leedahay daaweynta kansarka ugxan-sidaha iyo platinum iyo kansarka kale ee ugxan-sidaha iyo kansarka naasaha.Kansarka, kansarka mindhicirka sare, unugyada yaryar iyo kansarka sambabada unugyada aan yareyn waxay leeyihiin aragti wanaagsan.

 

Isticmaalka

Isticmaal 1: Botanicals-ka-hortagga burooyinka ballaaran ee kansarka ugxan-sidaha, kansarka naasaha, iwm.

Isticmaal 2: botanicals-ka-hortagga burooyinka ballaaran ee daaweynta kansarka ugxan-sidaha, kansarka naasaha iyo cudurrada kale.

Isticmaal 3: Daawooyinka lidka-tumorka.Daawaynta kansarka naasaha ee metastatic iyo kansarka ugxan-sidaha metastatic.Botanicals-ka-hortagga burooyinka ballaaran ee daaweynta kansarka ugxan-sidaha, kansarka naasaha iyo cudurrada kale.

Isticmaal 4: Daawo waxtar leh oo ka hortagga burooyinka;waxay kuxirantahay gobolka N-terminal ee β-tubulin, waxay kor u qaadaa microtubule hore oo xasiloon, waxay ka hortagtaa depolymerization, waxay ka hortagtaa kala qaybinta unugyada caadiga ah iyo dabinka marxaladda G2 / M ee wareegga unugyada.

Isticmaalka 5: Daawada lidka ku ah microtubule, ka hortagga depolymerization iyada oo kor u qaadeysa polymerization tubulin, ilaalinta xasilloonida tuubada, iyo joojinta mitosis unugga.

 

 


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