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Ganirelix Acetate Peptide API

Sharaxaad Gaaban:

Magaca: Ganirelix Acetate

Lambarka CAS: 123246-29-7

Qaaciddada molecular: C80H113ClN18O13

Miisaanka unugyada: 1570.34


Faahfaahinta Alaabta

Tags Product

Faahfaahinta Alaabta

Magaca Ganirelix Acetate
Lambarka CAS 123246-29-7
qaacidada molecular C80H113ClN18O13
Miisaanka molecular 1570.34

La mid ah

Ac-DNal-DCpa-DPal-Ser-Tyr-DHar(Et2)-Leu-Har(Et2)-Pro-DAla -NH2;Ganirelixum;ganirelix Acetate;GANIRELIX;Ganirelix Acetate USP/EP/

Sharaxaada

Ganirelix waa xarun decapeptide synthetic, iyo cusbada acetate, Ganirelix acetate waa gonadotropin-sii daynta hormoonka (GnRH) antagonist.Tixda amino acid waa: Ac-D-2Nal-D-4Cpa-D-3Pal-Ser-Tyr-D-HomoArg(9,10-Et2)-Leu-L-HomoArg(9,10-Et2)-Pro- D- Ala-NH2.Inta badan bukaan-socod ahaan, waxaa loo adeegsadaa haweenka lagu caawiyo tignoolajiyada taranka ee la xakameeyey barnaamijyada kicinta ugxan-sidaha si looga hortago heerka ugu sarreeya hoormoonka luteining-ka iyo in lagu daweeyo cilladaha bacriminta sababtan awgeed.Daroogadu waxay leedahay sifooyinka falcelinta xun xun, heerka uurka sare iyo muddada daawaynta gaaban, oo uu leeyahay faa'iidooyin cad marka la barbar dhigo daawooyinka la mid ah ee dhaqanka kiliinikada.

Falka dawooyinka

Sii daynta garaaca wadnaha ee hoormoonka sii daaya gonadotropin (GnRH) waxay kicisaa isku-dhafka iyo dheecaanka LH iyo FSH.Inta jeer ee garaaca wadnaha LH ee bartamaha iyo wejiyada dambe ee follicular waa qiyaastii 1 saac.garaaca wadnaha ayaa ka muuqda kor u kaca ku meel gaadhka ah ee serum LH.Inta lagu jiro xilliga caadada badhtamaha, siidaynta wayn ee GnRH waxay sababtaa kor u kaca LH.Koritaanka LH ee dhexdhexaadka ah wuxuu kicin karaa dhowr jawaabo nafsiyeed, oo ay ku jiraan: ugxansidaha, oocyte meiotic resumption, iyo samaynta corpus luteum.Sameynta luteum corpus waxay keentaa in heerka serum progesterone uu kordho, halka heerarka estradiol hoos u dhaco.Ganirelix acetate waa GnRH antagonist kaas oo si tartan ah u xannibaya soo-dhoweeyayaasha GnRH ee gonadotrophs pituitary iyo dariiqooyinka beddelka ee xiga.Waxay soo saartaa xannibaad degdeg ah, dib-u-noqosho ah ee dheecaanka gonadotropin.Saamaynta xannibaadda ganirelix acetate ee dheecaanka pituitary LH ayaa ka xoog badnaa tan FSH.Ganirelix acetate waxay ku guuldareysatay inay keento sii deynta ugu horeysa ee gonadotropins endogenous, oo la socota antagonism.Soo kabashada dhamaystiran ee heerarka LH pituitary iyo FSH ayaa dhacay 48 saacadood gudahood ka dib markii ganirelix acetate la joojiyay.


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