Magac | Eptifibibatide |
Lambarka CAS | 188627-80-7 |
Qaaciddada molika | C35h49n11o9s2 |
Miisaanka Moleculal | 831.96 |
Tirada EINECS | 641-366-7 |
Cucid | 1.60 ± 0.1 g / cm3 (la saadaaliyay) |
Xaaladaha kaydinta | Ku xidhan qalalan, ku keydi qaboojiyaha, ka yar -15 ° C |
Eptifibiyatidateecateecateecateecateecateteeacetates; eptifibibatide, mpa-har-harada-sm-sms-nh2, Mpahargdwpc-NH2, MPAHArgdwpc-NH2, Eptifiin; eptifibibatide; n6- ((aminomimi. Telethyl) -N2- ((3-Mercatto-1-Oxyfropyl-L-Lysylylcyl-L-trylyl-l-cysteyl-l-cysteropyde-l-cysterofyde-l-cysterogrid-re-cys-restrafrod-sm-cys) (isbarbardhigga 'Mpa1-CEYS6).
Etifibiid (Dhex-dhexaad) waa platettoptide platettoptide platelett 'glycoptotein gelcoprotein IIB / IIIIA Askagaganka' Plateritor ', kaas oo xannibay isku-darka platet iyo dhiig-xireyaasha iyadoo la xakameynayo dariiqa ugu dambeeya ee caadiga ah ee isku-darka platelet ee isku-darka platelet. Marka la barbar dhigo antibody-ka monoclonal abciximab, eptifibibatide wuxuu leeyahay xoog xoog leh oo jihooyin ah oo gaar ah iyo gaar ah oo loogu talagalay GPIB / III-daada jiritaanka hal-ka-beddelka amino acid ee amino-ka-xisbiga ah oo lagu beddelo arginine. Sidaa darteed, waa inay yeelato saameyn ku-daweynta wanaagsan ee daaweynta ku-dhexgalka ee cudurka choratery chonary syndrome. Daawooyinka platestet-ka ee Glcoprotein IIB / IIIIA Daawooyinka Antianortor-ka ayaa la soo saaray wax badan, oo hadda waxaa jira 3 nooc oo diyaarin ah oo lagu isticmaali karo taliska caalamiga ah, Abciximab, Eptifibibatide iyo Tirofifibanka. ). Khibrad yar ayaa ka jirta adeegsiga plateletprotein gpib / III-soo-nooleynta Shiinaha, daroogada la heli karo sidoo kale aad ayey u xadidan yihiin. Hal daroogo oo keliya, Trirofiban Hydrochloride, ayaa suuqa saaran. Sidaa darteed, waa platelet cusub oo glycoprotein IIB. / IIIIA Riptor Askarto waa lama huraan. Eptifibibatide gudaha ah waa badeecad ku dayasho mudan oo ay soo saartay badeecadaha bayoolaji ee Chengdu Sinro Coloy Sing., Ltd.
Kala-saaridda Dawooyinka Isku-darka Isku-darka
Daawooyinka isku-darka daroogada ee ka hortagga daroogada ayaa loo qaybin karaa saddex qaybood: 1. Cyclooxoxegalgeganse-1 (cox-1) xakameeyayaasha, sida asbiriin. 2. La'aanta isku-darka platelet ee uu sababay adenosine diphosphate (ADP), sida Cloperogel, sida ABCUGELEL, TICTIFIBIMOD, ETTIFIBIBID, EPTIFIBIIDE, EPTIBAN, EPT. Intaas waxaa dheer, waxaa jira prostagland ep3 Xaraashka soo-saareyaasha soo-saareyaasha, qaybaha kiimikada ee cusub ee isku-dhafka ah iyo soosaarka wax ku oolka ah ee ka soo baxa daawada Shiinaha ee caadiga ah.