Magac | DAPTOMYCIN |
Lambarka CAS | 103060-53-3 |
Qaaciddada molika | C72h101n17o26 |
Miisaanka Moleculal | 1620.67 |
Tirada EINECS | 600-389-2 |
Dhibcaha dhalaalaya | 202-204 ° C |
Point karkaraya | 2078.2 ± 65.0 ° C (saadaaliyay) |
Cucid | 1.45 ± 0.1 g / cm3 (saadaaliyay) |
Tooska Flash | 87 ℃ |
Xaaladaha kaydinta | Ku xidhan qalalan, ku keydi qaboojiyaha, hoosta -20 ° C |
Xaraash | Methanol: soluble5mg / ml |
Isutirka aashitada | (PKA) 4.00 ± 0.10 (la saadaaliyay) |
Qaab | budo |
Midab | Midab la'aan si huruud ah |
N- [n- (1-oxodechyl) -l-trp-d-asn-l-as-try-l-ser-l-gl-g-gl-g-gl-g-gl-r-gl-r-gl-r-gl-r-gl-r-gl-r-gl-r-gl-r-gl-r-gl-r-gl-r-gl-r-gl-r-gl-r-gl-r-gl-r-gl-r-gl-r-gl-r-gl-r-gl-r-gl-d-gl-r-gl-r-gl-r-gl-r-gl-d-gl-r-gl-r-gl-r-gl-r-gl-d-glu. - 4- (2-ameer-l-l-ye-l-by-l-by. ; Ecyl) -l-tryphophyl-d-aspartranyl-l-αyylylllycylcyl-l-sparttrulyl-d-αylllycyl-d-sparttrulllycyl-l-meheryl- α-spartrullllycyl-d-αyll-sl- (3R) -3-methyl-α- Glutamyl-α, 2-Dianino-ye-benzenutanobuid (13-4) lactomebutanoAninenocid (13-4) LaktonebutanoCutanocid (DAPTOme; DAPTYINE; DAPTYINE;
Antibiyootigyada Diptomycin waa antibiyootig isku dhafan oo lagu dhajiyo Wax ka beddelashada astaamaha xuubka cytoplasmic-ka ayaa carqaladeyn kara xuubka xuubka bakteeriyada siyaabo badan oo si dhakhso ah u dila bakteeriyada garaacista. Ka sokow awooda ay u leedahay in lagu dhaqmo bakteeriyada naxdinta leh ee ku habboon ee bakteeriyada ku habboon, DAPTOMYCIN waxay aad ugu muhimsan tahay dhibaatooyinka go'doonsan ee muujisay caabbinta methicillin, vancomycin, iyo zromycin. Waxay leedahay nashaad awood leh, oo hantidaasi waxay aad ugu muhiim u leedahay saameynno caafimaad oo aad u muhiim ah bukaannada si xun u xanuunsan. Cudurka oof wareenka eosinophilic waa cudur dhif ah oo aad u khatar ah oo leh astaamo ay ka mid yihiin qandho, qufac, neefsashada oo ku qabata, iyo neefsashada oo adkaata.
DAPTOMYCIN waxay leedahay waxqabad wanaagsan oo ka dhan ah bakteeriyada u adkeysta ee diinta u adkeysta, sida micnaha = 0.06-0.5 μg Mic = 0.0625 ~ 1μg / ml oo ah bakteeriyada, micni = 0.12 ~ 0.5μg / ml ee loo yaqaan 'antibilococcuspus epidermides', micni = ml = ml / ml) 0.5 ~ 1μg / ml, iyo ML-ka ee loo yaqaan 'aaladda' aaladda meteococcus u adkaysata antibiyootikada glycopeptis waa 1 ~ 2μg / ml.