Melanotan 1waa analoogga peptide synthetic eeα-MSH (alfa-melanocyte hormoonka kicinta). Waxay ku shaqeysaaDhaqdhaqaaqa melanocortin-1 reseptors (MC1R)kicinwax soo saarka melanin, bixinta dabiiciga ahmidabka maqaarkaiyoilaalinta sawir-qaadista.
Waxay ahaydloo oggolaaday daawaynta erythropoietic protoporphyria (EPP)-cilad naadir ah oo keenta dareen xad dhaaf ah oo iftiinka qoraxda ah. Melanotan 1 waxay caawisaa korodhkadulqaadka iftiinka UV, dhimofalcelinta phototoxic, iyo kor u qaadidadifaaca maqaarka ee waxyeellada UV-ku keeno.
XulashoMC1R agonist
Kordheysawax soo saarka eumelanin
Bixiyailaalinta qorraxda dabiiciga ah
TaageeroDayactirka DNA-da iyo ka-hortagga caabuqa
Suuragal u ahvitiligo, ka hortagga kansarka maqaarkaiyomidabaynta qurxinta
Lagu dhex baaraygabowga ka-hortaggaiyodaawaynta maqaarka
Nadiifin sare ≥99%
Waji adag oo peptide synthesis (SPPS)
Heerarka wax soo saarka ee GMP
Sahayda la qiyaasi karo: R&D ilaa heerar ganacsi